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This specific coordination geometry creates a stable yet bioavailable structure that maintains the copper ion in an optimal oxidation state for biological activity

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8.3 Buccal/sublingual delivery Buccal and sublingual delivery avoids GI degradation and partially avoids first-pass hepatic metabolism (venous drainage from these regions partially bypasses the portal circulation)

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10.1210/jc.2013-1029 102

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Pajares et al

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